SCHANEBERG, BRIAN T.1, WENDY L. APPLEQUIST2*, and IKHLAS A. KHAN1. 1National Center for Natural Products Research, Thad Cochran Research Center, The University of Mississippi, University, MS 38677; 2Missouri Botanical Garden, Applied Research Dept., P. O. Box 299, St. Louis, MO 63166-0299. - Is wild ginger toxic? Aristolochic acid content of North American species of Aristolochiaceae.
Chronic use of traditional herbal remedies containing
Aristolochia species (Aristolochiaceae) has been linked to
kidney failure and possibly cancer in humans, attributable to
aristolochic acid content. Asarum canadense (wild ginger) is
believed to contain aristolochic acids and has been banned from
commerce; however, wild ginger has a long history of safe folk use as
food and medicine, and numerous books for the public describe it as
edible. We sampled rhizomes from across its U.S. range, as well as the
rhizomes of other North American species of Aristolochiaceae, and
surveyed them for the presence of aristolochic acids I and II (AA I
and AA II) by HPLC. AA I and II were present in significant quantities
(maximum values of 0.39% and 0.66% respectively) in
Aristolochia species and Hexastylis arifolia. AA I alone
was detected in all samples of Asarum canadense and in minute
quantities in Asarum caudatum, though not in Asarum
wagneri. Concentrations in A. canadense were highly
variable, in one instance reaching 0.037% of dry weight. The highest
amounts were found in small populations under environmental pressure;
also, concentrations were higher in samples from the northeastern U.S.
and North Carolina than in those from the upper Midwest and South
Carolina. It is possible that long-term consumption of material from
high-AA populations would pose some risk of harm to susceptible
individuals. Pending better understanding of safe dosage limits and
the distribution of chemical races, a conservative approach to food
safety suggests that consumption of Asarum canadense should not
be encouraged in field guides or botany classes.
Key words: Aristolochiaceae, aristolochic acid, Asarum canadense, herbal medicine, Hexastylis